SCHEMBL5011747

SCHEMBL5011747

Cc1cccc(C(=O)N2N(Cc3ccc(C(C)(C)C)cc3)C(=O)OC23CCCCC3)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.40
HPGD P15428 1/20 0.40
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 1/20 0.37
OPRM1 P35372 2/20 0.37
OPRK1 P41145 1/20 0.37
ELANE P08246 1/20 0.37
SERPINE1 P05121 1/20 0.36
CYP2C9 P11712 2/20 0.36
OPRD1 P41143 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
PARG Q86W56 1/20 0.35
CCR9 P51686 1/20 0.35
CASP1 P29466 1/20 0.35
CASP8 Q14790 1/20 0.35
GABRD O14764 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011835 0.91 CYP1A2 (0.43) KCNK3HPGDLMNAALDH1A1CYP2C9
SCHEMBL5016329 0.89 CHRM2 (0.43) HPGDLMNAKMT2AALDH1A1OPRK1
SCHEMBL5011651 0.78 CHRM2 (0.44) LMNAKMT2AALDH1A1
SCHEMBL1086619 0.74 ALDH1A1 (0.46) HPGDKMT2AALDH1A1GABRDGABRA1
SCHEMBL5011879 0.73 KMT2A (0.38) HPGDLMNAKMT2AALDH1A1OPRM1
SCHEMBL5015148 0.73 LMNA (0.45) LMNAKMT2AALDH1A1ELANECYP2C9
SCHEMBL5015165 0.70 ATM (0.47) HPGDLMNAKMT2AALDH1A1CYP1A2
SCHEMBL5011708 0.70 CYP1A2 (0.45) HPGDLMNAKMT2AALDH1A1CYP1A2
SCHEMBL5011764 0.67 HTT (0.44) HPGDLMNAKMT2AALDH1A1
SCHEMBL1086170 0.65 EPHX2 (0.46) HPGDALDH1A1CYP2C9CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed