SCHEMBL5012782

SCHEMBL5012782

O=C1OC2(CCN(C(=O)c3ccc([N+](=O)[O-])cc3Cl)CC2)CN1Cc1ccc(SC(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.39
POLB P06746 3/20 0.39
LMNA P02545 5/20 0.38
KMT2A Q03164 1/20 0.38
MAPT P10636 8/20 0.37
SMN1; SMN2 Q16637 5/20 0.37
RAB9A P51151 2/20 0.37
GAA P10253 1/20 0.36
KCNK2 O95069 1/20 0.35
KCNK10 P57789 1/20 0.35
TP53 P04637 1/20 0.35
HTT P42858 2/20 0.35
NPC1 O15118 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GALR3 O60755 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5015186 0.90 SLC6A9 (0.43) ALDH1A1POLBLMNAKMT2AMAPT
SCHEMBL5015178 0.87 MAPT (0.47) ALDH1A1POLBLMNAKMT2AMAPT
SCHEMBL1086868 0.86 ALDH1A1 (0.41) ALDH1A1POLBLMNAKMT2AMAPT
SCHEMBL5016300 0.83 SLC6A9 (0.43) ALDH1A1POLBLMNAKMT2AMAPT
SCHEMBL1086411 0.82 ALDH1A1 (0.40) ALDH1A1POLBLMNAKMT2AMAPT
SCHEMBL1086551 0.81 TACR1 (0.42) KMT2ANPC1
SCHEMBL1086300 0.79 HTT (0.38) ALDH1A1POLBLMNAMAPTSMN1; SMN2
SCHEMBL1086423 0.79 TACR2 (0.39)
SCHEMBL1086626 0.78 ALDH1A1 (0.41) ALDH1A1POLBLMNAKMT2AMAPT
SCHEMBL1086255 0.78 ALDH1A1 (0.41) ALDH1A1POLBLMNAKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed