SCHEMBL5012784

SCHEMBL5012784

OC1(C(c2ccc(Oc3ncccn3)cc2)C(c2ccc(OC(F)(F)F)cc2)c2ccc(OC(F)(F)F)cc2)CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 8/20 0.39
MMP3 P08254 2/20 0.39
MMP1 P03956 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP13 P45452 1/20 0.39
MMP14 P50281 1/20 0.39
PDE5A O76074 1/20 0.37
PDE1A P54750 1/20 0.37
PDE3A Q14432 1/20 0.37
RXRA P19793 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
SLC6A2 P23975 8/20 0.36
NR1I2 O75469 1/20 0.35
MMP10 P09238 1/20 0.35
KCNH2 Q12809 1/20 0.35
SLC6A4 P31645 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5012781 0.89 PDE2A (0.38) PDE2AMMP3MMP1MMP9MMP8
SCHEMBL645639 0.78 SLC6A2 (0.40) PDE2ASLC6A2SLC6A4
SCHEMBL646801 0.74 SLC6A2 (0.43) PDE2AMMP3MMP1MMP9MMP8
SCHEMBL646388 0.71 KCNH2 (0.48) MMP3MMP1MMP9MMP8MMP13
SCHEMBL648546 0.69 RXRA (0.35) PDE2AMMP3MMP1MMP9MMP8
SCHEMBL647940 0.65 KCNH2 (0.48) MMP3MMP1MMP9MMP8MMP13
SCHEMBL31469761 0.65 SCN10A (0.37) MMP3MMP1MMP9MMP8MMP13
SCHEMBL5237277 0.65 DRD2 (0.54) MMP3MMP1MMP9MMP8MMP13
SCHEMBL14893597 0.65 NR1I2 (0.72) PDE2AMMP3MMP1MMP9MMP8
SCHEMBL3543085 0.62 EPHX1 (0.48) PDE2ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673083-A4 N-SUBSTITUTED AZACYCLES BAYER CROPSCIENCE AG (DE) 2008-12-17 EP disclosed
EP-1673083-A2 N-SUBSTITUTED AZACYCLES FMC CORPORATION (US) 2006-06-28 EP disclosed
WO-2005036961-A2 N-SUBSTITUTED AZACYCLES FMC CORPORATION (US) 2005-04-28 WO disclosed