SCHEMBL5013447

SCHEMBL5013447

COc1ccc([N+](=O)[O-])cc1CN1NC2(CCC(OC(=O)NC(C)c3cccc4ccccc34)CC2)OC1=O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PNKP Q96T60 3/20 0.41
TACR1 P25103 1/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
EDNRA P25101 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
TRPV1 Q8NER1 1/20 0.34
GAA P10253 1/20 0.34
ANO1 Q5XXA6 1/20 0.34
ANO2 Q9NQ90 1/20 0.34
GNRHR P30968 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4262148 0.77 PNKP (0.39) PNKPTACR1MEN1KMT2AEDNRA
SCHEMBL5015167 0.73 ALDH1A1 (0.40) TACR1MEN1KMT2AGAAGNRHR
SCHEMBL18375356 0.63 ALDH1A1 (0.46) MEN1KMT2ATRPV1GAALMNA
SCHEMBL29408478 0.63 ALDH1A1 (0.46) MEN1KMT2ATRPV1GAALMNA
SCHEMBL7932004 0.63 MEN1 (0.51) MEN1KMT2A
SCHEMBL7763963 0.63 PDE4A (0.40) MEN1KMT2AEDNRA
SCHEMBL7767275 0.63 PDE4A (0.40) MEN1KMT2AEDNRA
SCHEMBL7995664 0.62 PDE4B (0.41) MEN1KMT2AROCK2ROCK1
SCHEMBL8007232 0.62 PDE4B (0.41) MEN1KMT2AROCK2ROCK1
SCHEMBL7765376 0.62 EDNRA (0.41) MEN1KMT2AEDNRAROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed