SCHEMBL5014169

SCHEMBL5014169

CC(C)CCNc1cccc(Oc2ccc([N+](=O)[O-])c(N(C)C(=O)OC(C)(C)C)c2)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 2/20 0.36
POLB P06746 2/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
NPY5R Q15761 1/20 0.35
SIRT5 Q9NXA8 1/20 0.35
MMP13 P45452 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
NCOA1 Q15788 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33
NPC1 O15118 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4447217 0.86 MEN1 (0.40) GHSRKMT2AMEN1NPY5RMMP13
SCHEMBL3245632 0.83 MEN1 (0.42) POLBKMT2AMEN1MMP13ALDH1A1
SCHEMBL4453688 0.83 CETP (0.36) GHSRKMT2ANPY5RMMP13ALDH1A1
SCHEMBL27782513 0.81 SIRT5 (0.42) GHSRSIRT5MMP13ALDH1A1HTT
SCHEMBL6543839 0.81 MAPT (0.40) GHSRCYP2C19NPY5RMMP13ALDH1A1
SCHEMBL6544430 0.81 MMP13 (0.42) CYP2C19NPY5RMMP13ALDH1A1
SCHEMBL3487106 0.80 HSD17B1 (0.44) KMT2AMEN1ALDH1A1HTTMAPT
SCHEMBL3487759 0.80 MAPT (0.42) GHSRPOLBKMT2AMEN1ALDH1A1
SCHEMBL3488461 0.80 DHODH (0.38) KMT2AMEN1HTTMAPT
SCHEMBL6543697 0.79 MAPT (0.38) MMP13ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1982718-A1 ANTI-CANCER PHARMACEUTICAL COMPOSITION Daiichi Sankyo Company, Limited (JP) 2008-10-22 EP disclosed