SCHEMBL5014390

SCHEMBL5014390

CC1CN(c2c(CO)cc(-c3nnc(-c4ccccc4Cl)s3)c(F)c2F)CC(C)O1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.41
NPSR1 Q6W5P4 2/20 0.41
KDM4E B2RXH2 6/20 0.38
HIF1A Q16665 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37
HTT P42858 1/20 0.37
HPGD P15428 3/20 0.35
TDP1 Q9NUW8 1/20 0.35
GUSB P08236 1/20 0.35
MTOR P42345 2/20 0.35
HSD17B10 Q99714 2/20 0.34
RAB9A P51151 2/20 0.34
PIK3R1 P27986 1/20 0.34
PIK3CA P42336 1/20 0.34
NPC1 O15118 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
TP53 P04637 1/20 0.34
PKM P14618 1/20 0.34
CASP3 P42574 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5015619 0.91 HRH3 (0.37) ALDH1A1NPSR1KDM4EHRH3HTT
SCHEMBL5014366 0.88 ALDH1A1 (0.43) ALDH1A1NPSR1KDM4EHTTHPGD
SCHEMBL5012713 0.84 PIK3R1 (0.35) ALDH1A1NPSR1KDM4EHRH3HTT
SCHEMBL5015616 0.83 ALDH1A1 (0.39) ALDH1A1NPSR1KDM4EHIF1AHRH3
SCHEMBL5012716 0.82 PIK3R1 (0.34) ALDH1A1NPSR1KDM4EHTTHPGD
SCHEMBL5133875 0.82 PIK3R1 (0.34) ALDH1A1NPSR1KDM4EHTTHPGD
SCHEMBL5012742 0.81 PIK3R1 (0.34) ALDH1A1NPSR1KDM4EHRH3HTT
SCHEMBL5015657 0.81 PIK3R1 (0.34) ALDH1A1NPSR1KDM4EHTTHPGD
SCHEMBL5014333 0.81 PIK3R1 (0.36) ALDH1A1NPSR1KDM4EHTTHPGD
SCHEMBL5014337 0.78 KDM4E (0.35) ALDH1A1KDM4EHTTHPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888597-A2 ANTIBACTERIAL AGENTS Warner-Lambert Company LLC (US) 2008-02-20 EP disclosed
WO-2006120563-A2 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2006-11-16 WO disclosed