SCHEMBL5014395

SCHEMBL5014395

CC(C)(C)c1ccc(C2=NOC3(CCCCC3)N2OC(=O)Nc2ccccc2Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GLA P06280 1/20 0.43
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
FAAH O00519 1/20 0.38
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CHRM3 P20309 1/20 0.36
GAA P10253 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
BDKRB1 P46663 1/20 0.35
TRPV1 Q8NER1 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
MAPK14 Q16539 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5015752 0.82 LMNA (0.43) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL5012941 0.78 SMN1; SMN2 (0.36) RAB9ANPC1ALDH1A1L3MBTL1FAAH
SCHEMBL5010991 0.74 TRPV1 (0.41) RAB9ANPC1FAAHTP53MAPT
SCHEMBL16175602 0.74 ATM (0.43) RAB9ANPC1ALDH1A1GLAATM
SCHEMBL5054681 0.69 TRPV1 (0.58) TRPV1
SCHEMBL5125820 0.67 ALDH1A1 (0.45) RAB9ANPC1ALDH1A1GLAATM
SCHEMBL16175697 0.65 TRPM8 (0.39) RAB9ANPC1ATML3MBTL1MEN1
SCHEMBL5014557 0.64 CHRM3 (0.40) KMT2ACHRM3MAPT
SCHEMBL5014339 0.63 KMT2A (0.39) L3MBTL1FAAHKMT2ACHRM3
SCHEMBL5014399 0.63 CHRM3 (0.39) RAB9ANPC1MEN1KMT2ACHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888596-A1 SUBSTITUTED SPIRO COMPOUNDS AND THEIR USE FOR PRODUCING PAIN-RELIEF MEDICAMENTS Grünenthal GmbH (DE) 2008-02-20 EP claimed
WO-2006122770-A1 SUBSTITUTED SPIRO COMPOUNDS AND THEIR USE FOR PRODUCING PAIN-RELIEF MEDICAMENTS Grünenthal GmbH (DE) 2006-11-23 WO claimed