SCHEMBL5015339

SCHEMBL5015339

COc1ccccc1-c1cc(Cl)cc(NC(=O)O)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 7/20 0.60
ADORA1 P30542 2/20 0.55
ADORA2A P29274 3/20 0.51
ADORA2B P29275 2/20 0.49
HSP90AA1 P07900 2/20 0.48
HSP90AB1 P08238 1/20 0.48
ATR Q13535 1/20 0.46
DCTPP1 Q9H773 1/20 0.46
HSD17B10 Q99714 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
ALOX15 P16050 1/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4210224 0.82 APLNR (0.54) ADORA3ADORA1SMN1; SMN2MEN1MAPT
SCHEMBL4206294 0.80 HSP90AA1 (0.51) ADORA3ADORA1HSP90AA1HSP90AB1DCTPP1
SCHEMBL4204970 0.79 ADORA3 (0.51) ADORA3ADORA1ADORA2AHSP90AA1HSP90AB1
SCHEMBL4268096 0.78 ADORA1 (0.55) ADORA3ADORA1ADORA2AADORA2BSMN1; SMN2
Trifluoroacetic Acid SCHEMBL4200702 0.74 HSP90AA1 (0.51) ADORA3ADORA1ADORA2AHSP90AA1HSP90AB1
SCHEMBL4206708 0.73 HSP90AA1 (0.44) ADORA3ADORA1HSP90AA1HSP90AB1ATR
SCHEMBL4490553 0.72 HSP90AA1 (0.58) ADORA3ADORA1HSP90AA1HSP90AB1HSD17B10
SCHEMBL16965029 0.70 S1PR2 (0.44) ADORA3SMN1; SMN2MEN1MAPTRAB9A
SCHEMBL2468801 0.69 HSP90AA1 (0.54) ADORA3ADORA1ADORA2AHSP90AA1HSP90AB1
SCHEMBL26877045 0.69 HSP90AA1 (0.49) ADORA3ADORA1HSP90AA1HSP90AB1DCTPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1921066-A1 PYRIDYLPHENOL COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed