SCHEMBL5016765

SCHEMBL5016765

Cn1cncc1C(O)c1ccc2nc(Cl)nc(-c3cccc(Cl)c3)c2c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FNTA P49354 6/20 0.46
FNTB P49356 6/20 0.46
IDO1 P14902 1/20 0.44
PGGT1B P53609 6/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
CSNK2A2 P19784 1/20 0.37
CSNK2B P67870 1/20 0.37
MAT2A P31153 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5655017 0.81 FNTA (0.38) FNTAFNTBIDO1PGGT1BKDM4E
SCHEMBL6009561 0.81 FNTA (0.49) FNTAFNTBIDO1PGGT1B
SCHEMBL5543925 0.80 FNTA (0.60) FNTAFNTBIDO1PGGT1B
SCHEMBL7087571 0.79 IDO1 (0.40) FNTAFNTBIDO1PGGT1B
SCHEMBL7090215 0.79 FNTA (0.48) FNTAFNTBIDO1PGGT1B
SCHEMBL5026990 0.77 CSNK2A2 (0.45) FNTAFNTBIDO1PGGT1BKDM4E
SCHEMBL16632803 0.76 RORC (0.59)
SCHEMBL6010464 0.75 FNTA (0.60) FNTAFNTBIDO1PGGT1B
SCHEMBL6010160 0.75 FNTA (0.78) FNTAFNTB
SCHEMBL7093092 0.75 FNTA (0.44) FNTAFNTBIDO1PGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322650-B1 FARNESYL TRANSFERASE INHIBITING 6-HETEROCYCLYLMETHYL QUINOLINE AND QUINAZOLINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2008-09-24 EP disclosed
US-7196094-B2 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinoline and quinazoline derivatives JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-27 US disclosed
US-20030207887-A1 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinoline and quinazoline derivatives JANSSEN PHARMACEUTICA N.V. (BE) 2003-11-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030207887-A1 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinoline and quinazoline derivatives FNTA, FNTB, RCE1 FNTA 1/4885FNTB 2/4885IDO1 2867/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.