SCHEMBL5020165

SCHEMBL5020165

Bc1c(O)ccc2nc(C#N)ccc12

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSB P07858 2/20 0.43
SOS2 Q07890 1/20 0.41
NQO1 P15559 1/20 0.39
ESR1 P03372 5/20 0.33
ESR2 Q92731 5/20 0.33
ESRRB O95718 1/20 0.33
ESRRA P11474 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745771 0.79 ESR1 (0.51) CTSBSOS2NQO1ESR1ESR2
SCHEMBL7941665 0.75 SOS2 (0.50) CTSBSOS2NQO1ESR1ESR2
SCHEMBL5181894 0.75 SOS2 (0.56) CTSBSOS2NQO1ESR1ESR2
SCHEMBL5020169 0.73 MALT1 (0.34) CTSBNQO1
SCHEMBL13271162 0.69 CTSB (0.50) CTSBSOS2NQO1ESR1ESR2
SCHEMBL15413744 0.68 CYP3A4 (0.48) SOS2NQO1KDM4EALDH1A1
SCHEMBL30236776 0.68 CYP3A4 (0.48) SOS2NQO1KDM4EALDH1A1
SCHEMBL13291191 0.67 SOS2 (0.50) CTSBSOS2NQO1ESR1ESR2
SCHEMBL1996656 0.67 MAPT (0.57) SOS2NQO1KDM4EALDH1A1
SCHEMBL16372364 0.66 SOS2 (0.48) CTSBSOS2NQO1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064943-A2 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed