SCHEMBL5020169

SCHEMBL5020169

Bc1c(C(=O)C(F)(F)F)ccc2nc(C#N)ccc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 1/20 0.34
CAMKK2 Q96RR4 2/20 0.33
PLA2G2D Q9UNK4 1/20 0.33
NQO1 P15559 1/20 0.33
MLYCD O95822 1/20 0.32
ABL1 P00519 1/20 0.32
MAP2K2 P36507 1/20 0.32
CSNK1A1 P48729 1/20 0.32
CLK2 P49760 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
CDK5 Q00535 1/20 0.32
ACVR1 Q04771 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
DYRK1B Q9Y463 1/20 0.32
CTSB P07858 2/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8778585 0.84 CAMKK2 (0.33) MALT1CAMKK2PLA2G2DNQO1ABL1
SCHEMBL5020167 0.74 PLA2G2D (0.32) PLA2G2DMLYCD
SCHEMBL16914971 0.65 L3MBTL1 (0.44) CAMKK2NQO1PDE4APDE4BPDE4C
SCHEMBL16915197 0.65 NQO1 (0.41) CAMKK2NQO1PDE4APDE4BPDE4C
SCHEMBL31253334 0.65 SOS2 (0.41) CAMKK2CTSBMAPK1
SCHEMBL31324958 0.65 SOS2 (0.41) CAMKK2CTSBMAPK1
SCHEMBL838145 0.65 ALDH1A1 (0.41) CAMKK2CTSB
SCHEMBL25873382 0.64 NQO1 (0.40) NQO1CTSB
SCHEMBL8745729 0.64 NOTUM (0.39) MALT1NQO1CTSBPDE4APDE4B
SCHEMBL25585924 0.63 NAPRT (0.43) CAMKK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064943-A2 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed