SCHEMBL5020180

SCHEMBL5020180

CCOC(=O)NCc1cccc(-c2ccc(S(=O)(=O)NC(C)(C)C3CN=NN3)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.43
ALOX15 P16050 1/20 0.40
LMNA P02545 1/20 0.39
MMP1 P03956 2/20 0.38
MMP2 P08253 2/20 0.38
MMP3 P08254 2/20 0.38
MMP7 P09237 2/20 0.38
MMP10 P09238 2/20 0.38
MMP9 P14780 2/20 0.38
MMP8 P22894 2/20 0.38
MMP12 P39900 2/20 0.38
MMP14 P50281 2/20 0.38
MMP13 P45452 1/20 0.38
HDAC1 Q13547 1/20 0.37
ADAMTS4 O75173 3/20 0.36
NMT1 P30419 5/20 0.36
TSHR P16473 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5020184 0.91 BRD4 (0.43) MMP1MMP2MMP3MMP7MMP10
SCHEMBL5020143 0.90 MMP8 (0.39) MMP1MMP2MMP3MMP7MMP10
SCHEMBL8777128 0.76 GAA (0.45) GAAALOX15LMNAMMP1MMP2
SCHEMBL5020142 0.68 MMP2 (0.43) MMP1MMP2MMP3MMP7MMP10
SCHEMBL8777638 0.68 MMP2 (0.40) MMP1MMP2MMP3MMP7MMP10
SCHEMBL4906501 0.68 PADI3 (0.38) GAAMMP1MMP2MMP3MMP7
SCHEMBL6478104 0.67 TSHR (0.50) GAAHDAC1TSHRCYP2C19CYP2D6
SCHEMBL8777624 0.67 BRD4 (0.41) MMP1MMP2MMP3MMP7MMP10
SCHEMBL5020145 0.67 NMT1 (0.37) MMP1MMP2MMP3MMP7MMP10
SCHEMBL7788580 0.66 TSHR (0.67) GAAALOX15LMNAHDAC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064943-A2 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed