SCHEMBL5020775

SCHEMBL5020775

Cc1ccccc1NC(=O)/C=C/c1ccc(NS(=O)(=O)c2cccc3ccccc23)cc1

nearest known ligand 0.78

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.78
MMP1 P03956 4/20 0.56
MMP2 P08253 4/20 0.56
MMP9 P14780 4/20 0.56
EGFR P00533 1/20 0.56
TSHR P16473 1/20 0.52
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14629549 0.90 HDAC1 (0.63) HDAC1MMP1MMP2MMP9EGFR
SCHEMBL5020626 0.88 HDAC1 (1.00) HDAC1TSHR
SCHEMBL5047586 0.84 HDAC1 (1.00) HDAC1TSHR
SCHEMBL5020747 0.82 HDAC1 (0.78) HDAC1TSHR
SCHEMBL20657293 0.76 HDAC1 (0.60) HDAC1MMP1MMP2MMP9EGFR
N-O-Tolylcinnamamide SCHEMBL2593754 0.74 MMP1 (1.00) MMP1MMP2MMP9EGFRMAOA
N-O-Tolylcinnamamide SCHEMBL15902545 0.74 MMP1 (1.00) MMP1MMP2MMP9EGFRMAOA
N-O-Tolylcinnamamide SCHEMBL29844171 0.74 MMP1 (1.00) MMP1MMP2MMP9EGFRMAOA
N-O-Tolylcinnamamide SCHEMBL2593756 0.74 MMP1 (1.00) MMP1MMP2MMP9EGFRMAOA
SCHEMBL4471817 0.74 KDM4E (0.57) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE43343-E1 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-05-01 US disclosed