SCHEMBL5020747

SCHEMBL5020747

CC(=O)/C=C/c1ccc(NS(=O)(=O)c2cccc3ccccc23)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 10/20 0.78
TSHR P16473 1/20 0.61
PGR P06401 1/20 0.54
RORA P35398 1/20 0.53
RORC P51449 1/20 0.53
NR1H2 P55055 1/20 0.53
NR1H4 Q96RI1 1/20 0.53
ALDH1A1 P00352 1/20 0.52
HTT P42858 1/20 0.52
PFKFB3 Q16875 1/20 0.52
HCRTR1 O43613 1/20 0.50
BRD4 O60885 1/20 0.48
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5047586 0.88 HDAC1 (1.00) HDAC1TSHRBRD4HDAC3HDAC4
SCHEMBL5020763 0.83 HDAC1 (0.82) HDAC1TSHRBRD4
SCHEMBL5020775 0.82 HDAC1 (0.78) HDAC1TSHR
SCHEMBL5020749 0.81 HDAC1 (0.80) HDAC1ALDH1A1HTT
SCHEMBL5020626 0.80 HDAC1 (1.00) HDAC1TSHR
SCHEMBL14629549 0.80 HDAC1 (0.63) HDAC1TSHRPGRRORARORC
SCHEMBL5020753 0.78 HDAC1 (0.78) HDAC1PGRALDH1A1HDAC3HDAC4
SCHEMBL3261087 0.77 TSHR (0.71) HDAC1TSHRPGRRORARORC
SCHEMBL16785737 0.77 TSHR (0.67) HDAC1TSHRPGRRORARORC
SCHEMBL812673 0.76 TSHR (0.74) HDAC1TSHRPGRRORARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE43343-E1 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-05-01 US disclosed