SCHEMBL5021141

SCHEMBL5021141

NC1CCCc2cc(CO)c(CO)cc21

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.40
ESR1 P03372 3/20 0.33
ESR2 Q92731 3/20 0.33
OPRD1 P41143 2/20 0.32
IGF1R P08069 1/20 0.32
ALOX15 P16050 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1726880 0.76 OPRD1 (0.45) ACHEESR1ESR2OPRD1
SCHEMBL4517111 0.76 OPRD1 (0.45) ACHEESR1ESR2OPRD1
SCHEMBL1726878 0.76 OPRD1 (0.45) ACHEESR1ESR2OPRD1
SCHEMBL11164638 0.76 IGF1R (0.53) ACHEIGF1RALOX15ADRA2AADRA2B
SCHEMBL15109677 0.72 ACHE (0.40) ACHEOPRD1
SCHEMBL15109754 0.72 HTR2A (0.41) ACHEESR1ESR2OPRD1
SCHEMBL28170162 0.70 ACHE (0.43) ACHEADRA2AADRA2BADRA2CADRA1D
SCHEMBL3535473 0.69 KDM1A (0.45) ACHEESR1ESR2
SCHEMBL2803692 0.69 ACHE (0.51) ACHEESR1ESR2
SCHEMBL8274690 0.69 ESR1 (0.55) ACHEESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120115850-A1 SUBSTITUTED ARYLAMINE COMPOUNDS AND METHODS OF TREATMENT BECKER OREN (IL) 2012-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120115850-A1 SUBSTITUTED ARYLAMINE COMPOUNDS AND METHODS OF TREATMENT HTR6, HTR2A, HTR3B ACHE 1589/4885ESR1 1353/4885ESR2 502/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.