SCHEMBL5024129

SCHEMBL5024129

CN(C)CCN(C(=O)[C@H]1CC[C@H](CN(C)c2ncc(Br)cn2)CC1)C1CC1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.34
CCNK O75909 2/20 0.33
CDK12 Q9NYV4 2/20 0.33
LSS P48449 1/20 0.31
ALDH1A1 P00352 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5028487 0.88 GRIN2B (0.35) GRIN2BCDK12ALDH1A1PKM
SCHEMBL5025673 0.80 TAS2R14 (0.38) GRIN2BALDH1A1
SCHEMBL5025675 0.80 TAS2R14 (0.38) GRIN2BALDH1A1
SCHEMBL20772888 0.78 DAO (0.36) GRIN2BLSS
SCHEMBL5024145 0.74 KMT2A (0.40) GRIN2BALDH1A1PKM
SCHEMBL5024150 0.74 KMT2A (0.40) GRIN2BALDH1A1PKM
SCHEMBL14174989 0.72 L3MBTL1 (0.40) ALDH1A1
SCHEMBL5024054 0.71 HTT (0.54) GRIN2B
SCHEMBL5024052 0.71 HTT (0.54) GRIN2B
SCHEMBL5024111 0.70 PLG (0.35) LSSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7442791-B2 Aminoalkylamide substituted cyclohexyl derivatives HOFFMANN-LA ROCHE INC. (US) 2008-10-28 US disclosed
EP-1667962-A1 AMINOALKYLAMIDE SUBSTITUTED CYCLOHEXYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-06-14 EP disclosed
WO-2005028427-A1 AMINOALKYLAMIDE SUBSTITUTED CYCLOHEXYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-03-31 WO disclosed
US-20050065210-A1 Aminoalkylamide substituted cyclohexyl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2005-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065210-A1 Aminoalkylamide substituted cyclohexyl derivatives LSS, CYP51A1, CYP46A1 GRIN2B 4512/4885CCNK 194/4885CDK12 1571/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.