SCHEMBL5027115

SCHEMBL5027115

COC[C@@H]1C[C@H](N(C)C(C)C)CC[C@@H]1N(Cc1ccccc1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.43
RORC P51449 2/20 0.39
CYP2D6 P10635 2/20 0.38
KCNH2 Q12809 2/20 0.38
UBE2M P61081 5/20 0.37
DCUN1D1 Q96GG9 5/20 0.37
CTSD P07339 1/20 0.37
REN P00797 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
MMP13 P45452 1/20 0.36
OPRM1 P35372 2/20 0.36
CCR5 P51681 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5027117 1.00 CCR2 (0.43) CCR2RORCCYP2D6KCNH2UBE2M
SCHEMBL5027120 1.00 CCR2 (0.43) CCR2RORCCYP2D6KCNH2UBE2M
SCHEMBL5031820 0.75 CCR2 (0.39) CCR2RORCCYP2D6KCNH2MEN1
SCHEMBL5031949 0.71 SLC6A2 (0.38) CCR2RORCCYP2D6KCNH2MEN1
SCHEMBL5033700 0.70 CCR2 (0.44) CCR2CYP2D6KCNH2RENCCR5
SCHEMBL5029381 0.70 SLC6A4 (0.38) CCR2RORCCYP2D6KCNH2
SCHEMBL5027340 0.69 CCR2 (0.53) CCR2CYP2D6KCNH2CCR5
SCHEMBL21359110 0.69 CTSD (0.50) DCUN1D1CTSDOPRM1MEN1KMT2A
SCHEMBL3370759 0.68 AGER (0.55) DCUN1D1CTSDOPRM1MEN1KMT2A
SCHEMBL21359174 0.68 CTSD (0.49) CTSDOPRM1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7378409-B2 Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-27 US disclosed