SCHEMBL5027399

SCHEMBL5027399

COc1cc(OCCC2CCCCN2)ccc1N

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
CYP3A4 P08684 1/20 0.45
CHRNB4 P30926 3/20 0.45
CHRNA3 P32297 3/20 0.45
CHEK2 O96017 1/20 0.45
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HIF1A Q16665 1/20 0.42
PHLPP2 Q6ZVD8 1/20 0.42
HPGD P15428 1/20 0.41
LTA4H P09960 5/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5025845 0.96 CHRNB4 (0.49) ALDH1A1CYP3A4CHRNB4CHRNA3CHEK2
SCHEMBL11449248 0.91 CHRNB4 (0.50) CHRNB4CHRNA3CHEK2MEN1KMT2A
SCHEMBL11457361 0.87 CHRNB4 (0.54) CHRNB4CHRNA3CHEK2MEN1KMT2A
SCHEMBL11449154 0.84 LTA4H (0.50) CHEK2CYP1A2CYP2D6CYP2C19SMN1; SMN2
SCHEMBL11715221 0.82 LTA4H (0.53) CHEK2LTA4H
SCHEMBL11449447 0.82 CYP1A2 (0.48) CHRNB4CHRNA3CYP1A2CYP2D6CYP2C19
SCHEMBL11716280 0.81 LTA4H (0.50) CHRNB4CHRNA3CHEK2LTA4H
SCHEMBL6073607 0.81 CHRNB4 (0.47) CHRNB4CHRNA3CHEK2CYP1A2CYP2D6
SCHEMBL6628961 0.81 CHRNB4 (0.51) CHRNB4CHRNA3CHEK2CYP1A2CYP2D6
SCHEMBL6600614 0.81 NFE2L2 (0.60) CHEK2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919892-A2 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORPORATION (US) 2008-05-14 EP disclosed
WO-2007027527-A2 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORPORATION (US) 2007-03-08 WO disclosed