SCHEMBL5031160

SCHEMBL5031160

NC(=O)CC(=O)N(c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
PTGIR P43119 3/20 0.38
PTGDR Q13258 2/20 0.38
KCNN4 O15554 1/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NR3C2 P08235 1/20 0.37
AGTR2 P50052 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1136766 0.83 CYP3A4 (0.48) KMT2A
SCHEMBL8242543 0.82 HTT (0.42) ALDH1A1PTGIRPTGDRESR1ESR2
SCHEMBL10272760 0.81 POLQ (0.49) ALDH1A1
SCHEMBL16111874 0.81 SMN1; SMN2 (0.43) ALDH1A1NPC1POLBHTTRAB9A
SCHEMBL29063529 0.81 CYP2C9 (0.43) ALDH1A1PTGIRPTGDRNPC1POLB
SCHEMBL8405808 0.80 KIF11 (0.44) ALDH1A1
SCHEMBL830792 0.80 ALDH1A1 (0.59) ALDH1A1NPC1POLBHTTRAB9A
SCHEMBL10364096 0.79 HDAC3 (0.44) ALDH1A1ESR1ESR2
SCHEMBL8243336 0.78 ALDH1A1 (0.41) ALDH1A1PTGIRPTGDRPOLBHTT
SCHEMBL5808336 0.77 KCNN4 (0.45) ALDH1A1KCNN4ESR1ESR2NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896395-B1 MODIFIED MALONATE DERIVATIVES MERCK SHARP & DOHME (US) 2015-07-15 EP disclosed
EP-1896395-A2 MODIFIED MALONATE DERIVATIVES Merck & Co., Inc. (US) 2008-03-12 EP disclosed
WO-2007002248-A2 MODIFIED MALONATE DERIVATIVES MERCK & CO., INC. (US) 2007-01-04 WO disclosed