SCHEMBL5808336

SCHEMBL5808336

NC(=O)N(c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 5/20 0.45
ALDH1A1 P00352 1/20 0.45
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
TSHR P16473 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
S100A4 P26447 1/20 0.39
MAPK14 Q16539 1/20 0.39
NR3C2 P08235 1/20 0.38
SLC22A2 O15244 1/20 0.38
SLC22A1 O15245 1/20 0.38
SLC22A3 O75751 1/20 0.38
PLAU P00749 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27958929 0.98 KCNN4 (0.43) KCNN4ALDH1A1CES2CES1ESR1
SCHEMBL6037507 0.90 ACHE (0.50) KCNN4ALDH1A1TSHRMAPK14
SCHEMBL11729778 0.88 BCL2L1 (0.57) CES2CES1ESR1ESR2TSHR
SCHEMBL2237446 0.81 CA2 (0.57) CA1CA2
SCHEMBL753482 0.81 S100A4 (0.33) KCNN4ALDH1A1ESR1ESR2TSHR
SCHEMBL11845019 0.79 KCNN4 (0.43) KCNN4ALDH1A1CES2CES1CA1
SCHEMBL65464 0.78 ALDH1A1 (0.44) ALDH1A1TSHRPLAU
SCHEMBL11417635 0.78 ESR1 (0.43) ALDH1A1ESR1ESR2CA1CA2
SCHEMBL4589533 0.77 ALDH1A1 (0.47) KCNN4ALDH1A1CES2CES1
SCHEMBL320721 0.77 KCNN4 (0.42) KCNN4ALDH1A1CES2CES1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006130426-A2 MODULATORS OF CCR-5 ACTIVITY KEMIA, INC. (US) 2006-12-07 WO claimed
US-4698444-A 1,1-bis(p-fluorophenyl)urea PFIZER INC. (US) 1987-10-06 US claimed
US-4477669-A Processes and intermediates useful in the preparation of flutroline PFIZER INC. (US) 1984-10-16 US claimed
EP-0082658-A2 Processes and intermediates useful in the preparation of flutroline PFIZER INC. (US) 1983-06-29 EP claimed
WO-2006130426-A2 MODULATORS OF CCR-5 ACTIVITY KEMIA, INC. (US) 2006-12-07 WO disclosed
US-4698444-A 1,1-bis(p-fluorophenyl)urea PFIZER INC. (US) 1987-10-06 US disclosed
US-4698444-A 1,1-bis(p-fluorophenyl)urea PFIZER INC. (US) 1987-10-06 US disclosed
US-4698444-A 1,1-bis(p-fluorophenyl)urea PFIZER INC. (US) 1987-10-06 US disclosed
US-4568748-A 2-Carbobenzoxy-8-fluoro-5-(p-fluorophenyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole PFIZER INC. (US) 1986-02-04 US disclosed
US-4568748-A 2-Carbobenzoxy-8-fluoro-5-(p-fluorophenyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole PFIZER INC. (US) 1986-02-04 US disclosed
US-4477669-A Processes and intermediates useful in the preparation of flutroline PFIZER INC. (US) 1984-10-16 US disclosed
US-4477669-A Processes and intermediates useful in the preparation of flutroline PFIZER INC. (US) 1984-10-16 US disclosed
US-4467090-A Compound, 8-fluoro-5-(p-fluorophenyl)-2-[4-(p-fluorophenyl)-4-hydroxybutyryl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole PFIZER INC. (US) 1984-08-21 US disclosed
EP-0082658-A3 PROCESSES AND INTERMEDIATES USEFUL IN THE PREPARATION OF FLUTROLINE PFIZER INC. (US) 1984-06-06 EP disclosed
EP-0082658-A2 Processes and intermediates useful in the preparation of flutroline PFIZER INC. (US) 1983-06-29 EP disclosed
EP-0082658-A2 Processes and intermediates useful in the preparation of flutroline PFIZER INC. (US) 1983-06-29 EP disclosed