SCHEMBL5032145

SCHEMBL5032145

NC(=O)CCCc1c[nH]nc1-c1nc(NCc2ccccc2)c2ncn([C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.58
TP53 P04637 1/20 0.56
SLC29A1 Q99808 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
PGK1 P00558 3/20 0.53
PGK2 P07205 3/20 0.53
ADORA2A P29274 4/20 0.52
ADORA1 P30542 3/20 0.52
NT5E P21589 3/20 0.52
ADORA2B P29275 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5034055 0.83 ADORA1 (0.60) ADORA3SLC29A1ADORA2AADORA1NT5E
SCHEMBL5038188 0.82 ADORA3 (0.59) ADORA3TP53SLC29A1TDP1PGK1
SCHEMBL6582374 0.81 ADORA3 (0.63) ADORA3TP53SLC29A1TDP1PGK1
SCHEMBL6584541 0.81 ADORA3 (0.64) ADORA3TP53SLC29A1TDP1PGK1
SCHEMBL5034054 0.81 ADORA3 (0.59) ADORA3TP53SLC29A1TDP1PGK1
SCHEMBL5040344 0.81 ADORA3 (0.59) ADORA3TP53SLC29A1TDP1PGK1
SCHEMBL5035415 0.81 ADORA3 (0.59) ADORA3TP53SLC29A1TDP1PGK1
SCHEMBL5397146 0.80 ADORA3 (0.58) ADORA3TP53SLC29A1TDP1PGK1
SCHEMBL4136495 0.79 ADORA3 (0.61) ADORA3TP53SLC29A1TDP1ADORA2A
SCHEMBL4136498 0.79 ADORA3 (0.61) ADORA3TP53SLC29A1TDP1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881991-A1 A1 ADENOSINE RECEPTOR AGONISTS CV THERAPEUTICS, INC. (US) 2008-01-30 EP claimed
WO-2006125211-A1 A1 ADENOSINE RECEPTOR AGONISTS CV THERAPEUTICS, INC. (US) 2006-11-23 WO claimed
EP-1881991-A1 A1 ADENOSINE RECEPTOR AGONISTS CV THERAPEUTICS, INC. (US) 2008-01-30 EP disclosed
WO-2006125211-A1 A1 ADENOSINE RECEPTOR AGONISTS CV THERAPEUTICS, INC. (US) 2006-11-23 WO disclosed