SCHEMBL5035001

SCHEMBL5035001

CCN(C)C(=O)Oc1cnc(N(C(=O)c2ccc(Cl)cc2Cl)c2ccc(OC)c(OC)c2)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.41
TSHR P16473 2/20 0.39
GAA P10253 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
FLT1 P17948 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
QPCT Q16769 3/20 0.34
MCOLN3 Q8TDD5 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HSP90AA1 P07900 1/20 0.33
BCHE P06276 1/20 0.33
MAOA P21397 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032683 0.93 CYP3A4 (0.37) CYP3A4TSHRGAANPSR1FLT1
SCHEMBL5034781 0.93 CYP3A4 (0.42) CYP3A4TSHRGAANPSR1FLT1
SCHEMBL5041456 0.90 CYP3A4 (0.48) CYP3A4GAANPSR1ALDH1A1MAPT
SCHEMBL5035233 0.89 CYP3A4 (0.38) CYP3A4TSHRGAANPSR1FLT1
SCHEMBL5032514 0.88 CYP3A4 (0.43) CYP3A4TSHRGAANPSR1FLT1
SCHEMBL5039337 0.85 CYP3A4 (0.34) CYP3A4TSHRGAANPSR1FLT1
SCHEMBL5036072 0.83 CYP3A4 (0.44) CYP3A4GAANPSR1ALDH1A1MAPT
SCHEMBL5032512 0.83 CYP3A4 (0.40) CYP3A4TSHRGAANPSR1FLT1
SCHEMBL5032529 0.82 CYP3A4 (0.43) CYP3A4TSHRGAANPSR1FLT1
SCHEMBL14190190 0.82 FLT1 (0.41) CYP3A4TSHRFLT1FLT4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP claimed