SCHEMBL5039337

SCHEMBL5039337

COc1ccc(N(C(=O)c2ccc(Cl)cc2Cl)c2ncc(OC(=O)N(CCO)C(C)(C)C)s2)cc1OC

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.34
FLT1 P17948 1/20 0.34
FLT4 P35916 1/20 0.34
KDR P35968 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
TSHR P16473 1/20 0.33
PYGL P06737 1/20 0.33
SCD O00767 1/20 0.32
GAA P10253 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
QPCT Q16769 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.31
CSF1R P07333 2/20 0.31
NR1H4 Q96RI1 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5035170 0.88 CYP3A4 (0.36) CYP3A4FLT1FLT4KDRIRAK4
SCHEMBL5034781 0.87 CYP3A4 (0.42) CYP3A4FLT1FLT4KDRTSHR
SCHEMBL5032683 0.85 CYP3A4 (0.37) CYP3A4FLT1FLT4KDRIRAK4
SCHEMBL5035001 0.85 CYP3A4 (0.41) CYP3A4FLT1FLT4KDRTSHR
SCHEMBL5035233 0.84 CYP3A4 (0.38) CYP3A4FLT1FLT4KDRTSHR
SCHEMBL5036081 0.81 CYP3A4 (0.35) CYP3A4FLT1FLT4KDRIRAK4
SCHEMBL14190190 0.79 FLT1 (0.41) CYP3A4FLT1FLT4KDRTSHR
SCHEMBL5032642 0.78 CYP3A4 (0.41) CYP3A4GAANPSR1
SCHEMBL5035234 0.78 ALDH1A1 (0.41) CYP3A4FLT1FLT4KDRTSHR
SCHEMBL5032512 0.77 CYP3A4 (0.40) CYP3A4FLT1FLT4KDRIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP claimed