SCHEMBL5035010

SCHEMBL5035010

CCN(CCN(C)C)C(=O)Oc1csc(N(C(=O)c2ccc(Cl)cc2Cl)c2ccc(OC)c(OC)c2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
TSHR P16473 2/20 0.37
HCRTR2 O43614 5/20 0.35
HCRTR1 O43613 3/20 0.35
ALDH1A1 P00352 2/20 0.34
FLT1 P17948 1/20 0.34
FLT4 P35916 1/20 0.34
KDR P35968 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TLR9 Q9NR96 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5039107 0.94 CYP3A4 (0.38) CYP3A4TSHRHCRTR2HCRTR1ALDH1A1
SCHEMBL5035949 0.94 CYP3A4 (0.42) CYP3A4TSHRHCRTR2HCRTR1ALDH1A1
SCHEMBL5032562 0.93 CRHBP (0.36) CYP3A4TSHRFLT1FLT4KDR
SCHEMBL5035235 0.92 CYP3A4 (0.45) CYP3A4ALDH1A1GAAMAPTHTT
SCHEMBL5032631 0.89 CYP3A4 (0.37) CYP3A4TSHRALDH1A1FLT1FLT4
SCHEMBL5041208 0.89 CYP3A4 (0.41) CYP3A4TSHRHCRTR2HCRTR1ALDH1A1
SCHEMBL5041489 0.86 CYP3A4 (0.41) CYP3A4TSHRALDH1A1GAAMAPT
SCHEMBL5039136 0.86 CYP3A4 (0.44) CYP3A4ALDH1A1HTTNPC1RAB9A
SCHEMBL5035948 0.86 CYP3A4 (0.40) CYP3A4TSHRALDH1A1FLT1FLT4
SCHEMBL5041385 0.86 CYP3A4 (0.46) CYP3A4ALDH1A1MAPTHTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP claimed