SCHEMBL5032562

SCHEMBL5032562

COc1ccc(N(C(=O)c2ccc(Cl)cc2Cl)c2nc(OC(=O)N(C)CCN(C)C)cs2)cc1OC

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 2/20 0.36
CRHR2 Q13324 2/20 0.36
CYP3A4 P08684 2/20 0.35
FLT1 P17948 1/20 0.35
FLT4 P35916 1/20 0.35
KDR P35968 1/20 0.35
HSP90AA1 P07900 1/20 0.34
TSHR P16473 1/20 0.34
HRH4 Q9H3N8 2/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
RAD52 P43351 1/20 0.33
IRAK4 Q9NWZ3 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032631 0.93 CYP3A4 (0.37) CRHBPCRHR2CYP3A4FLT1FLT4
SCHEMBL5035010 0.93 CYP3A4 (0.39) CRHBPCRHR2CYP3A4FLT1FLT4
SCHEMBL5036077 0.91 CYP3A4 (0.42) CYP3A4HRH4CYP11B1CYP11B2RAD52
SCHEMBL5035949 0.90 CYP3A4 (0.42) CYP3A4FLT1FLT4KDRTSHR
SCHEMBL5036040 0.88 LMNA (0.42) CYP3A4HSP90AA1MEN1KMT2A
SCHEMBL14190166 0.87 CYP3A4 (0.37) CRHBPCRHR2CYP3A4FLT1FLT4
SCHEMBL5039107 0.87 CYP3A4 (0.38) CYP3A4FLT1FLT4KDRTSHR
SCHEMBL5041489 0.87 CYP3A4 (0.41) CRHBPCRHR2CYP3A4TSHRCYP11B1
SCHEMBL5035948 0.85 CYP3A4 (0.40) CRHBPCRHR2CYP3A4FLT1FLT4
SCHEMBL5035235 0.84 CYP3A4 (0.45) CYP3A4CYP11B1CYP11B2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP claimed