SCHEMBL5032631

SCHEMBL5032631

CCCN(C)C(=O)Oc1csc(N(C(=O)c2ccc(Cl)cc2Cl)c2ccc(OC)c(OC)c2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.37
IRAK4 Q9NWZ3 2/20 0.37
CRHBP P24387 2/20 0.36
CRHR2 Q13324 2/20 0.36
TSHR P16473 1/20 0.36
FLT1 P17948 1/20 0.35
FLT4 P35916 1/20 0.35
KDR P35968 1/20 0.35
NPSR1 Q6W5P4 2/20 0.34
HSP90AA1 P07900 1/20 0.34
KMT2A Q03164 3/20 0.33
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HTT P42858 2/20 0.33
MEN1 O00255 2/20 0.33
MAPT P10636 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032562 0.93 CRHBP (0.36) CYP3A4IRAK4CRHBPCRHR2TSHR
SCHEMBL5034877 0.91 CYP3A4 (0.44) CYP3A4IRAK4KMT2AKDM4EL3MBTL1
SCHEMBL5035949 0.90 CYP3A4 (0.42) CYP3A4TSHRFLT1FLT4KDR
SCHEMBL5035010 0.89 CYP3A4 (0.39) CYP3A4IRAK4CRHBPCRHR2TSHR
SCHEMBL5041489 0.88 CYP3A4 (0.41) CYP3A4IRAK4CRHBPCRHR2TSHR
SCHEMBL5036040 0.88 LMNA (0.42) CYP3A4HSP90AA1KMT2AALDH1A1GAA
SCHEMBL5035199 0.87 CYP3A4 (0.39) CYP3A4IRAK4CRHBPCRHR2TSHR
SCHEMBL5039107 0.87 CYP3A4 (0.38) CYP3A4TSHRFLT1FLT4KDR
SCHEMBL5035948 0.86 CYP3A4 (0.40) CYP3A4CRHBPCRHR2TSHRFLT1
SCHEMBL5034908 0.85 CYP3A4 (0.43) CYP3A4KMT2AHTTMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP claimed