SCHEMBL5035284

SCHEMBL5035284

COc1ccc2c(c1)c(C(=O)N(C)C1CCN(C)CC1)cn2S(=O)(=O)c1ccc(OC)c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 17/20 0.53
ALDH1A1 P00352 1/20 0.46
CYP3A4 P08684 2/20 0.43
ADRA2A P08913 2/20 0.43
CYP2D6 P10635 2/20 0.43
ADRA2C P18825 2/20 0.43
CYP2C19 P33261 2/20 0.43
HTR2A P28223 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3759250 0.95 HTR6 (0.49) HTR6ALDH1A1CYP3A4ADRA2ACYP2D6
SCHEMBL3746693 0.92 HTR6 (0.58) HTR6ALDH1A1
Trifluoroacetic Acid SCHEMBL3754067 0.88 HTR6 (0.51) HTR6ALDH1A1
Trifluoroacetic Acid SCHEMBL3754269 0.87 HTR6 (0.49) HTR6ALDH1A1CYP3A4CYP2D6HTR2A
Trifluoroacetic Acid SCHEMBL3753593 0.78 HTR6 (0.49) HTR6ALDH1A1HTR2A
Trifluoroacetic Acid SCHEMBL3761902 0.75 HTR6 (0.40) HTR6CYP3A4ADRA2ACYP2D6ADRA2C
SCHEMBL3747271 0.73 ALDH1A1 (0.46) HTR6ALDH1A1
Trifluoroacetic Acid SCHEMBL3752797 0.70 AVPR1B (0.52) HTR6HTR2A
SCHEMBL3754250 0.70 FABP4 (0.58) HTR6ALDH1A1
SCHEMBL3749236 0.69 HTR6 (1.00) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1476151-B1 1-ARYLSULFONYL-3-SUBSTITUED INDOLE AND INDOLINE DERIVATES USEFUL IN THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ORGANON NV (NL) 2008-07-16 EP disclosed