SCHEMBL5036571

SCHEMBL5036571

CCCc1cc(-c2ccc(Cl)cc2)nc2c(OC(=O)Nc3cccc(S(N)(=O)=O)c3)cnn12

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 0.47
CA9 Q16790 9/20 0.47
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 2/20 0.45
CA1 P00915 8/20 0.44
CA12 O43570 7/20 0.44
MAPT P10636 1/20 0.42
CA5A P35218 1/20 0.40
PKM P14618 1/20 0.40
CA4 P22748 2/20 0.39
CA7 P43166 1/20 0.39
GLA P06280 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5034960 0.94 CA2 (0.48) CA2CA9KMT2AMEN1ALDH1A1
SCHEMBL5035314 0.93 KMT2A (0.39) CA2CA9KMT2AMEN1ALDH1A1
SCHEMBL5041510 0.88 CA2 (0.52) CA2CA9KMT2AMEN1ALDH1A1
SCHEMBL5034907 0.88 KIF18A (0.45) CA2CA9KMT2AKDM4EHTT
SCHEMBL5039326 0.86 KMT2A (0.40) CA2CA9KMT2AMEN1ALDH1A1
SCHEMBL5049382 0.86 CA2 (0.53) CA2CA9KMT2AMEN1ALDH1A1
SCHEMBL5039198 0.84 CA2 (0.48) CA2CA9KMT2AMEN1ALDH1A1
SCHEMBL5039328 0.84 CA2 (0.46) CA2CA9KMT2AMEN1ALDH1A1
SCHEMBL5035270 0.84 MAPK1 (0.54) CA2CA9KMT2AMEN1ALDH1A1
SCHEMBL5034946 0.82 RIPK2 (0.43) CA2CA9KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed