SCHEMBL5036948

SCHEMBL5036948

C=CCC(Cc1ccc(Cl)cc1)NC(C)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 8/20 0.51
MME P08473 2/20 0.42
PSMB5 P28074 1/20 0.41
ACE P12821 1/20 0.40
ROCK2 O75116 1/20 0.40
PRKACA P17612 1/20 0.40
RPS6KB1 P23443 1/20 0.40
IRAK1 P51617 1/20 0.40
PRKX P51817 1/20 0.40
LIMK1 P53667 1/20 0.40
PRKG2 Q13237 1/20 0.40
ROCK1 Q13464 1/20 0.40
PRKG1 Q13976 1/20 0.40
PKN2 Q16513 1/20 0.40
HIPK4 Q8NE63 1/20 0.40
AURKB Q96GD4 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
CSNK1G1 Q9HCP0 1/20 0.40
HTT P42858 1/20 0.39
CTSC P53634 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5036248 1.00 ACACB (0.51) ACACBMMEPSMB5ACEROCK2
SCHEMBL7615213 0.87 MME (0.46) ACACBMMEPSMB5ACEROCK2
SCHEMBL8481611 0.86 FPR2 (0.41) ACACBMMEPSMB5ACEROCK2
SCHEMBL5033815 0.85 CTRB1 (0.53) MME
SCHEMBL5043208 0.85 CTRB1 (0.53) MME
SCHEMBL5033810 0.85 CTRB1 (0.53) MME
SCHEMBL14195827 0.81 ACACB (0.56) ACACBMMEACEROCK2PRKACA
SCHEMBL8926162 0.80 HTT (0.45) MMEROCK2PRKACARPS6KB1IRAK1
SCHEMBL10051044 0.80 MME (0.50) ACACBMME
SCHEMBL10051046 0.80 MME (0.50) ACACBMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1889903-A1 Biocatalysts with amine acylase activity Novartis AG (CH) 2008-02-20 EP disclosed
EP-0954571-B1 BIOCATALYSTS WITH AMINE ACYLASE ACTIVITY NOVARTIS AG (CH) 2007-08-29 EP disclosed
US-6235516-B1 FROM RHODOCOCCUS GLOBERULUS, RHODOCOCCUS EQUI OR ARTHROBACTER AURESCENS NOVARTIS AG (CH) 2001-05-22 US disclosed
EP-0954571-A1 BIOCATALYSTS WITH AMINE ACYLASE ACTIVITY Novartis AG (CH) 1999-11-10 EP disclosed
WO-1997041214-A1 BIOCATALYSTS WITH AMINE ACYLASE ACTIVITY NOVARTIS AG (CH) 1997-11-06 WO disclosed