SCHEMBL5037644

SCHEMBL5037644

Oc1cccc(-c2ccc(Cl)cc2)c1.Oc1cccc(-c2cccc(Cl)c2)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 8/20 0.68
HSD17B2 P37059 7/20 0.68
CYP3A4 P08684 2/20 0.68
CYP2C9 P11712 2/20 0.68
TSHR P16473 1/20 0.61
ALOX5 P09917 2/20 0.60
ESR2 Q92731 3/20 0.55
TAAR1 Q96RJ0 1/20 0.53
CNR1 P21554 1/20 0.53
ESR1 P03372 3/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2B6 P20813 1/20 0.52
CYP2C19 P33261 1/20 0.52
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
MAOB P27338 2/20 0.49
ABL1 P00519 1/20 0.48
ABCB1 P08183 1/20 0.48
BCR P11274 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1028579 0.94 HSD17B1 (0.77) HSD17B1HSD17B2CYP3A4CYP2C9TSHR
SCHEMBL1029061 0.92 TSHR (0.73) HSD17B1HSD17B2CYP3A4CYP2C9TSHR
SCHEMBL1520884 0.87 TAAR1 (0.65) ALOX5ESR2TAAR1CNR1CYP1A2
SCHEMBL29776911 0.87 TAAR1 (0.65) ALOX5ESR2TAAR1CNR1CYP1A2
SCHEMBL5379998 0.85 ESR1 (0.70) HSD17B1HSD17B2CYP3A4CYP2C9TSHR
SCHEMBL29434858 0.85 ESR1 (0.70) HSD17B1HSD17B2CYP3A4CYP2C9TSHR
Phenol SCHEMBL28114880 0.83 TSHR (0.60) HSD17B1HSD17B2CYP3A4CYP2C9TSHR
SCHEMBL7898375 0.82 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2C9ESR2
SCHEMBL16394285 0.82 TAAR1 (0.71) ALOX5ESR2TAAR1CYP1A2MAOB
SCHEMBL31491189 0.82 TAAR1 (0.71) ALOX5ESR2TAAR1CYP1A2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957493-A1 8-AZABICYCLO[3.2.1]OCTANE DERIVATIVES USEFUL AS MONOAMINE REUPTAKE INHIBITORS N.V. Organon (NL) 2008-08-20 EP disclosed
WO-2007063071-A1 8-AZABICYCLO[3.2.1]OCTANE DERIVATIVES USEFUL AS MONOAMINE REUPTAKE INHIBITORS N.V. ORGANON (NL) 2007-06-07 WO disclosed