SCHEMBL5037832

SCHEMBL5037832

Cc1ccc(CNC(=O)Cc2cccc(CC(C)(C)NC[C@@H](O)c3ccc(O)c(NS(C)(=O)=O)c3)c2)cc1

nearest known ligand 0.89

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 19/20 0.89
CHRM3 P20309 1/20 0.62
ADRB3 P13945 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5037827 1.00 ADRB2 (0.89) ADRB2CHRM3ADRB3
SCHEMBL5037075 0.94 ADRB2 (1.00) ADRB2CHRM3ADRB3
SCHEMBL5037072 0.94 ADRB2 (1.00) ADRB2CHRM3ADRB3
SCHEMBL5034412 0.93 ADRB2 (0.86) ADRB2CHRM3ADRB3
SCHEMBL5034410 0.93 ADRB2 (0.86) ADRB2CHRM3ADRB3
SCHEMBL12305722 0.93 ADRB2 (0.90) ADRB2CHRM3
SCHEMBL5034534 0.93 ADRB2 (0.88) ADRB2CHRM3ADRB3
SCHEMBL5037020 0.93 ADRB2 (0.88) ADRB2CHRM3
SCHEMBL5034540 0.93 ADRB2 (0.88) ADRB2CHRM3ADRB3
SCHEMBL5037018 0.93 ADRB2 (0.88) ADRB2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7351742-B2 Sulfonamide derivatives for the treatment of diseases PFIZER INC. (US) 2008-04-01 US claimed
EP-1708992-B1 SULFONAMIDE DERIVATIVES FOR THE TREATMENT OF DISEASES PFIZER LTD (GB) 2007-08-08 EP claimed
US-20050171147-A1 Sulfonamide derivatives for the treatment of diseases PFIZER INC. 2005-08-04 US claimed
US-7351742-B2 Sulfonamide derivatives for the treatment of diseases PFIZER INC. (US) 2008-04-01 US disclosed
EP-1708992-B1 SULFONAMIDE DERIVATIVES FOR THE TREATMENT OF DISEASES PFIZER LTD (GB) 2007-08-08 EP disclosed
US-20050171147-A1 Sulfonamide derivatives for the treatment of diseases PFIZER INC. 2005-08-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171147-A1 Sulfonamide derivatives for the treatment of diseases SULT2A1, STS, SULT1A1 ADRB2 2148/4885CHRM3 1774/4885ADRB3 2520/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.