SCHEMBL5039082

SCHEMBL5039082

CC(C)(CO)NS(=O)(=O)c1cccc(NC(=O)Oc2cnn3c(C(F)F)cc(-c4ccc(Cl)cc4)nc23)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
KMT2A Q03164 2/20 0.49
HTT P42858 1/20 0.49
MAPK1 P28482 1/20 0.48
KIF18A Q8NI77 4/20 0.47
TP53 P04637 3/20 0.44
POLB P06746 2/20 0.44
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 3/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
THRB P10828 1/20 0.41
GLA P06280 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5039141 0.92 KDM4E (0.49) KDM4EKMT2AHTTMAPK1KIF18A
SCHEMBL5039327 0.90 KIF18A (0.47) KDM4EKMT2AHTTMAPK1KIF18A
SCHEMBL5041449 0.89 KIF18A (0.46) KDM4EKMT2AHTTMAPK1KIF18A
SCHEMBL5036074 0.89 KIF18A (0.46) KDM4EKMT2AHTTMAPK1KIF18A
SCHEMBL5046611 0.88 MAPK1 (0.58) KDM4EKMT2AHTTMAPK1KIF18A
SCHEMBL5041408 0.87 KIF18A (0.45) KDM4EKMT2AHTTKIF18A
SCHEMBL5034907 0.87 KIF18A (0.45) KDM4EKMT2AHTTMAPK1KIF18A
SCHEMBL5036170 0.87 KDM4E (0.44) KDM4EKMT2AHTTMAPK1KIF18A
SCHEMBL5035287 0.87 KDM4E (0.49) KDM4EKMT2AHTTMAPK1KIF18A
SCHEMBL5035270 0.86 MAPK1 (0.54) KDM4EKMT2AHTTMAPK1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed