SCHEMBL5040928

SCHEMBL5040928

O=C(ON(Cc1ccc(F)cc1)C1CCNCC1)C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.51
SLC6A4 P31645 9/20 0.47
SLC6A2 P23975 8/20 0.47
SLC6A3 Q01959 4/20 0.47
HTR2A P28223 3/20 0.44
DCUN1D1 Q96GG9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5037869 0.89 TACR1 (0.41) TACR1SLC6A4SLC6A2SLC6A3DCUN1D1
SCHEMBL5033623 0.87 ALDH1A1 (0.46) TACR1SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL5040988 0.87 HTR2C (0.47) TACR1SLC6A4SLC6A2HTR2ADCUN1D1
SCHEMBL5036146 0.86 SLC6A2 (0.51) TACR1SLC6A4SLC6A2SLC6A3DCUN1D1
SCHEMBL5040993 0.82 SLC6A4 (0.58) SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL5037787 0.81 SLC6A2 (0.49) SLC6A4SLC6A2SLC6A3
SCHEMBL5040950 0.75 SLC6A2 (0.36) SLC6A4SLC6A2SLC6A3
SCHEMBL5034052 0.74 SLC6A2 (0.43) SLC6A4SLC6A2SLC6A3
SCHEMBL20781111 0.72 TACR1 (0.59) TACR1SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL5140305 0.72 TACR1 (0.55) TACR1SLC6A4SLC6A2SLC6A3HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622914-A4 NEW PIPERIDINYLAMINO-THIENO 2,3-D PYRIMIDINE COMPOUNDS EPIX DELAWARE INC (US) 2008-03-12 EP disclosed
EP-1622914-A2 NEW PIPERIDINYLAMINO-THIENO 2,3-D PYRIMIDINE COMPOUNDS Predix Pharmaceuticals Holdings, Inc. (US) 2006-02-08 EP disclosed
WO-2004089312-A2 NEW PIPERIDINYLAMINO-THIENO[2,3-D] PYRIMIDINE COMPOUNDS PREDIX PHARMACEUTICALS HOLDINGS, INC. (US) 2004-10-21 WO disclosed