SCHEMBL5040993

SCHEMBL5040993

O=C(ON(Cc1ccc2ccccc2c1)C1CCNCC1)C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 20/20 0.58
SLC6A2 P23975 18/20 0.58
SLC6A3 Q01959 16/20 0.58
KCNH2 Q12809 6/20 0.56
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR7 P34969 1/20 0.45
HTR2B P41595 1/20 0.45
HTR3A P46098 1/20 0.45
HTR4 Q13639 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5036146 0.83 SLC6A2 (0.51) SLC6A4SLC6A2SLC6A3
SCHEMBL5040928 0.82 TACR1 (0.51) SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL5040988 0.82 HTR2C (0.47) SLC6A4SLC6A2HTR2AHTR2C
SCHEMBL5033623 0.82 ALDH1A1 (0.46) SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL5037869 0.81 TACR1 (0.41) SLC6A4SLC6A2SLC6A3
SCHEMBL5037787 0.78 SLC6A2 (0.49) SLC6A4SLC6A2SLC6A3
SCHEMBL5034052 0.74 SLC6A2 (0.43) SLC6A4SLC6A2SLC6A3
SCHEMBL5040950 0.70 SLC6A2 (0.36) SLC6A4SLC6A2SLC6A3
SCHEMBL28014872 0.70 ITGB3 (0.41) SLC6A4SLC6A2SLC6A3HTR2AHTR2C
Trifluoroacetic Acid SCHEMBL312779 0.70 SLC6A2 (0.68) SLC6A4SLC6A2SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622914-A4 NEW PIPERIDINYLAMINO-THIENO 2,3-D PYRIMIDINE COMPOUNDS EPIX DELAWARE INC (US) 2008-03-12 EP disclosed
EP-1622914-A2 NEW PIPERIDINYLAMINO-THIENO 2,3-D PYRIMIDINE COMPOUNDS Predix Pharmaceuticals Holdings, Inc. (US) 2006-02-08 EP disclosed
WO-2004089312-A2 NEW PIPERIDINYLAMINO-THIENO[2,3-D] PYRIMIDINE COMPOUNDS PREDIX PHARMACEUTICALS HOLDINGS, INC. (US) 2004-10-21 WO disclosed