SCHEMBL5040988

SCHEMBL5040988

O=C(ON(Cc1ccc(OC(F)(F)F)cc1)C1CCNCC1)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.47
EPHX1 P07099 1/20 0.45
SLC6A2 P23975 3/20 0.39
SLC6A4 P31645 3/20 0.39
TACR1 P25103 1/20 0.39
DCUN1D1 Q96GG9 1/20 0.39
SCN9A Q15858 1/20 0.38
GCGR P47871 3/20 0.38
HTR2A P28223 2/20 0.38
LSS P48449 1/20 0.38
GIPR P48546 1/20 0.37
CXCR3 P49682 1/20 0.37
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5033623 0.88 ALDH1A1 (0.46) SLC6A2SLC6A4TACR1DCUN1D1HTR2A
SCHEMBL5040928 0.87 TACR1 (0.51) SLC6A2SLC6A4TACR1DCUN1D1HTR2A
SCHEMBL5037869 0.86 TACR1 (0.41) SLC6A2SLC6A4TACR1DCUN1D1
SCHEMBL5040993 0.82 SLC6A4 (0.58) HTR2CSLC6A2SLC6A4HTR2A
SCHEMBL5036146 0.78 SLC6A2 (0.51) SLC6A2SLC6A4TACR1DCUN1D1
SCHEMBL5037787 0.75 SLC6A2 (0.49) SLC6A2SLC6A4
SCHEMBL5040950 0.72 SLC6A2 (0.36) SLC6A2SLC6A4
SCHEMBL5995736 0.71 SLC6A2 (0.73) SLC6A2SLC6A4
SCHEMBL5034052 0.71 SLC6A2 (0.43) SLC6A2SLC6A4
Trifluoroacetic Acid SCHEMBL5040982 0.71 HTR2C (0.58) HTR2CEPHX1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622914-A4 NEW PIPERIDINYLAMINO-THIENO 2,3-D PYRIMIDINE COMPOUNDS EPIX DELAWARE INC (US) 2008-03-12 EP disclosed
EP-1622914-A2 NEW PIPERIDINYLAMINO-THIENO 2,3-D PYRIMIDINE COMPOUNDS Predix Pharmaceuticals Holdings, Inc. (US) 2006-02-08 EP disclosed
WO-2004089312-A2 NEW PIPERIDINYLAMINO-THIENO[2,3-D] PYRIMIDINE COMPOUNDS PREDIX PHARMACEUTICALS HOLDINGS, INC. (US) 2004-10-21 WO disclosed