SCHEMBL5041539

SCHEMBL5041539

CS(=O)(=O)c1cccc(NC(=O)Oc2cnn3ccc(-c4ccc(C(F)(F)F)cc4)nc23)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.43
KCNH2 Q12809 1/20 0.41
EPHX2 P34913 2/20 0.40
RXFP1 Q9HBX9 2/20 0.39
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
PLK4 O00444 2/20 0.37
KIF18A Q8NI77 1/20 0.37
PTGS2 P35354 2/20 0.36
RIPK1 Q13546 1/20 0.36
SCN5A Q14524 2/20 0.36
MGLL Q99685 1/20 0.36
MAPK1 P28482 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
PTK2 Q05397 1/20 0.36
IDH2 P48735 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5035282 0.92 CA2 (0.46)
SCHEMBL5035097 0.89 LMNA (0.43) KCNH2RXFP1KDM4EHTTKMT2A
SCHEMBL5035013 0.86 KDM4E (0.46) NTRK1RXFP1KDM4EHTTKMT2A
SCHEMBL5032666 0.86 NTRK1 (0.44) NTRK1EPHX2RXFP1KDM4EHTT
SCHEMBL5041227 0.85 RXFP1 (0.48) NTRK1KCNH2RXFP1KDM4EHTT
SCHEMBL5039150 0.84 KDM4E (0.54) NTRK1KDM4EHTTKMT2AMAPK1
SCHEMBL5035007 0.83 NTRK1 (0.41) NTRK1EPHX2RXFP1KDM4EHTT
SCHEMBL5035086 0.80 CA2 (0.51) KMT2AMAPT
SCHEMBL5041442 0.79 KDM4E (0.45) RXFP1KDM4EHTTKMT2AMAPK1
SCHEMBL5035278 0.79 CA2 (0.44) KDM4EHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed