SCHEMBL5041565

SCHEMBL5041565

N=C(N)c1ccc(CNC(=O)C(N)c2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 2/20 0.62
ST14 Q9Y5Y6 1/20 0.58
F2 P00734 14/20 0.57
MASP2 O00187 3/20 0.57
F10 P00742 3/20 0.55
PRSS1 P07477 3/20 0.55
TMPRSS6 Q8IU80 2/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
F7 P08709 2/20 0.48
KLKB1 P03952 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5041567 1.00 TPSAB1 (0.62) TPSAB1ST14F2MASP2F10
Hydrochloric Acid SCHEMBL5041862 0.99 TPSAB1 (0.60) TPSAB1ST14F2MASP2F10
Hydrochloric Acid SCHEMBL5041868 0.99 TPSAB1 (0.60) TPSAB1ST14F2MASP2F10
Hydrochloric Acid SCHEMBL21995166 0.87 KMT2A (0.58) MEN1KMT2A
SCHEMBL4220537 0.85 KMT2A (0.55) MEN1KMT2A
Hydrochloric Acid SCHEMBL4205709 0.84 KMT2A (0.54) MEN1KMT2A
Hydrochloric Acid SCHEMBL4205714 0.84 KMT2A (0.54) MEN1KMT2A
SCHEMBL5047815 0.83 F2 (0.61) TPSAB1ST14F2MASP2F10
SCHEMBL5047819 0.83 F2 (0.61) TPSAB1ST14F2MASP2F10
SCHEMBL5042149 0.82 PKM (0.70) TPSAB1ST14F2MASP2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567498-B1 MANDELIC ACID DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-23 EP disclosed
EP-1567498-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-08-31 EP disclosed
WO-2004048335-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-06-10 WO disclosed