SCHEMBL5044188

SCHEMBL5044188

O=C(O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F.O=c1oc2cc(S)ccc2c(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.41
ESR2 Q92731 2/20 0.41
ERAP1 Q9NZ08 1/20 0.40
THRB P10828 1/20 0.37
KDM4E B2RXH2 3/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 1/20 0.37
STAT1 P42224 1/20 0.37
RAB9A P51151 1/20 0.37
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
POLB P06746 1/20 0.34
ATM Q13315 1/20 0.34
PLEC Q15149 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5044620 0.82 ESR1 (0.54) ESR1ESR2ERAP1KDM4EKMT2A
SCHEMBL6869907 0.73 THRB (0.44) ERAP1THRBKDM4EKMT2AALDH1A1
Biphenyl SCHEMBL27611650 0.73 PGR (0.44) ERAP1KDM4EKMT2AALDH1A1NPC1
Trifluoromethanesulfonic Acid SCHEMBL3521218 0.71 ERAP1 (0.39) ESR1ESR2ERAP1KDM4EKMT2A
SCHEMBL5041731 0.71 THRB (0.39) THRBKDM4EALDH1A1NPC1RAB9A
SCHEMBL31675834 0.69 ESR1 (0.82) ESR1ESR2ERAP1THRBKDM4E
SCHEMBL5082203 0.69 ESR1 (0.82) ESR1ESR2ERAP1THRBKDM4E
SCHEMBL3366067 0.67 ESR1 (0.88) ESR1ESR2ERAP1THRBKDM4E
SCHEMBL8934513 0.67 ESR1 (0.88) ESR1ESR2ERAP1THRBKDM4E
SCHEMBL1800595 0.65 CA1 (0.56) ESR1ESR2ERAP1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1481973-B1 HETEROCYCLE-BEARING ONIUM SALTS WAKO PURE CHEM IND LTD (JP) 2008-12-31 EP disclosed
EP-1953149-A2 A heterocycle-containing onium salt Wako Pure Chemical Industries, Ltd. (JP) 2008-08-06 EP disclosed
EP-1481973-A1 HETEROCYCLE-BEARING ONIUM SALTS Wako Pure Chemical Industries, Ltd. (JP) 2004-12-01 EP disclosed