SCHEMBL5044867

SCHEMBL5044867

CCCCCCCCCCCc1noc(-c2cccc(C([NH])Cc3cccc(-c4ccccc4)c3)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
NPC1 O15118 1/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
HPGD P15428 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HSD17B10 Q99714 1/20 0.47
SPHK2 Q9NRA0 10/20 0.45
SPHK1 Q9NYA1 10/20 0.45
CHRM2 P08172 3/20 0.40
CHRM4 P08173 3/20 0.40
CHRM5 P08912 3/20 0.40
CHRM1 P11229 3/20 0.40
CHRM3 P20309 3/20 0.40
NOTUM Q6P988 1/20 0.35
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5045817 0.92 ALDH1A1 (0.53) ALDH1A1KDM4ENPC1MAPTPKM
SCHEMBL5047736 0.92 ALDH1A1 (0.53) ALDH1A1KDM4ENPC1MAPTPKM
SCHEMBL5044424 0.86 ALDH1A1 (0.50) ALDH1A1KDM4ENPC1MAPTPKM
SCHEMBL5044858 0.82 ALDH1A1 (0.40) ALDH1A1KDM4ENPC1MAPTPKM
SCHEMBL1856445 0.81 ALDH1A1 (0.53) ALDH1A1KDM4ENPC1MAPTPKM
SCHEMBL5039878 0.80 ALDH1A1 (0.38) ALDH1A1KDM4ENPC1MAPTPKM
SCHEMBL6802901 0.79 ALDH1A1 (0.41) ALDH1A1KDM4ENPC1MAPTPKM
SCHEMBL5039990 0.78 SPHK1 (0.41) ALDH1A1KDM4ENPC1MAPTPKM
SCHEMBL5045783 0.78 PPARG (0.44) ALDH1A1KDM4ENPC1MAPTPKM
SCHEMBL1853630 0.77 ALDH1A1 (0.51) ALDH1A1KDM4ENPC1MAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732534-B1 USE OF METHYLENE AMIDE DERIVATIVES IN CARDIOVASCULAR DISORDERS SERONO LAB (CH) 2008-07-23 EP claimed
EP-1470102-A1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) Applied Research Systems ARS Holding N.V. (AN) 2004-10-27 EP disclosed
WO-2003064376-A1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2003-08-07 WO disclosed