SCHEMBL5045757

SCHEMBL5045757

CC(NC(=O)OC(C)(C)C)C(C)C(=O)N1CCN(c2ccc(Cl)cc2)C(C)(C)C1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 7/20 0.54
DRD2 P14416 5/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TRPA1 O75762 1/20 0.36
STS P08842 1/20 0.36
MMP14 P50281 1/20 0.36
ADAMTS5 Q9UNA0 1/20 0.36
MC4R P32245 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4497465 0.88 CCR1 (0.67) CCR1MEN1KMT2ATRPA1
SCHEMBL4497464 0.88 CCR1 (0.67) CCR1MEN1KMT2ATRPA1
SCHEMBL3943101 0.78 CCR1 (0.59) CCR1DRD2
SCHEMBL3943882 0.77 DRD2 (0.59) CCR1DRD2MEN1KMT2ASMN1; SMN2
SCHEMBL5050629 0.76 CCR1 (0.49) CCR1DRD2MEN1KMT2AHTT
SCHEMBL4504830 0.74 CCR1 (0.61) CCR1MEN1KMT2AMMP14ADAMTS5
SCHEMBL4504825 0.74 CCR1 (0.61) CCR1MEN1KMT2AMMP14ADAMTS5
SCHEMBL13606430 0.73 CCR1 (0.67) CCR1
SCHEMBL4507643 0.73 CCR1 (0.74) CCR1
SCHEMBL4507638 0.73 CCR1 (0.74) CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973880-A1 PIPERAZINYL DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Brystol-Myers Squibb Company (US) 2008-10-01 EP disclosed
WO-2007087585-A1 PIPERAZINYL DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2007-08-02 WO disclosed