SCHEMBL5048288

SCHEMBL5048288

O=C1[N]NC(=O)C(c2ccc(Cl)cc2)=C1c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.49
GSK3B P49841 6/20 0.39
RECQL P46063 2/20 0.39
NOTUM Q6P988 3/20 0.37
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
TSHR P16473 1/20 0.36
GSK3A P49840 1/20 0.36
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5769180 0.92 GCGR (0.46) PTGS2ALDH1A1KDM4EMAPTLMNA
SCHEMBL8001119 0.77 CYP1A2 (0.47) GSK3BKDM4EGAAMAPTLMNA
SCHEMBL3816794 0.68 GSK3B (0.67) PTGS2GSK3BGSK3A
SCHEMBL6111216 0.68 NOTUM (0.36) RECQLNOTUMALDH1A1KDM4EGAA
SCHEMBL6704189 0.65 PTGS2 (0.58) PTGS2GSK3BRECQLALDH1A1KDM4E
SCHEMBL3823878 0.64 PTGS2 (0.56) PTGS2GSK3BKDM4EGAAMAPT
SCHEMBL3820693 0.63 GSK3B (0.63) PTGS2GSK3BGSK3A
SCHEMBL10593567 0.63 CYP2D6 (0.39) PTGS2GSK3BRECQLNOTUMALDH1A1
SCHEMBL91966 0.63 PTGS2 (0.50) PTGS2GSK3BRECQLNOTUMALDH1A1
SCHEMBL3823556 0.62 GSK3B (0.54) PTGS2GSK3BGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891074-A1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS Brystol-Myers Squibb Company (US) 2008-02-27 EP disclosed
WO-2006138682-A1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-12-28 WO disclosed
EP-1697371-A1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS Bristol-Myers Squibb Company (US) 2006-09-06 EP disclosed
WO-2005063762-A1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-14 WO disclosed