SCHEMBL5049686

SCHEMBL5049686

C=CCOC(=O)CCC1CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.45
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
TSHR P16473 2/20 0.42
PKM P14618 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
EPHX2 P34913 1/20 0.36
ITGB3 P05106 5/20 0.35
ITGA2B P08514 5/20 0.35
TPSAB1 Q15661 1/20 0.35
TPSD1 Q9BZJ3 1/20 0.35
TPSG1 Q9NRR2 1/20 0.35
HTR4 Q13639 1/20 0.34
GNAI3 P08754 1/20 0.34
GNAO1 P09471 1/20 0.34
GNAI1 P63096 1/20 0.34
FAAH O00519 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19629 0.83 CASP1 (0.60) CASP1ALDH1A1GAATSHRTDP1
Hydrochloric Acid SCHEMBL15158064 0.79 CASP1 (0.44) CASP1ALDH1A1GAATSHRPKM
SCHEMBL14037434 0.78 TSHR (0.44) CASP1ALDH1A1GAATSHRPKM
Acetic Acid SCHEMBL28331584 0.78 CASP1 (0.58) CASP1ALDH1A1GAATSHRTDP1
SCHEMBL3597232 0.78 TDP1 (0.44) ALDH1A1GAATSHRPKMITGB3
Propionic Acid SCHEMBL13280009 0.77 CASP1 (0.60) CASP1ALDH1A1GAATSHRPKM
Hydrochloric Acid SCHEMBL2942254 0.77 GNAI3 (0.44) ALDH1A1GAAPKMITGB3ITGA2B
SCHEMBL8556452 0.75 GNAI3 (0.43) ALDH1A1ITGB3ITGA2BHTR4GNAI3
SCHEMBL23521223 0.75 ALDH1A1 (0.45) CASP1ALDH1A1GAATSHRPKM
SCHEMBL16649239 0.75 ALDH1A1 (0.42) CASP1ALDH1A1GAATSHRPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1988078-A1 Carboxamide derivatives of pyrrolidine, piperidine and hexahydroazepine for the treatment of thrombosis disorders Ortho-McNeil Pharmaceutical, Inc. (US) 2008-11-05 EP disclosed
CN-1286684-A Carboxamide derivs. of pyrrolidine, piperidine and hexahydroazepine for treatment of thrombosis disorders ORTHO PHARMA CORP (US) 2001-03-07 CN disclosed
EP-0923555-A1 CARBOXAMIDE DERIVATIVES OF PYRROLIDINE, PIPERIDINE AND HEXAHYDROAZEPINE FOR THE TREATMENT OF THROMBOSIS DISORDERS ORTHO PHARMACEUTICAL CORPORATION (US) 1999-06-23 EP disclosed
WO-1997041102-A1 CARBOXAMIDE DERIVATIVES OF PYRROLIDINE, PIPERIDINE AND HEXAHYDROAZEPINE FOR THE TREATMENT OF THROMBOSIS DISORDERS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-11-06 WO disclosed