SCHEMBL5056159

SCHEMBL5056159

O=C1OC2(CCCCC2)N(C(=O)c2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)N1Cc1ccc(SC(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR6 P46095 1/20 0.38
MAPT P10636 4/20 0.37
TRPC3 Q13507 2/20 0.37
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ACHE P22303 1/20 0.34
POLB P06746 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CCR1 P32246 3/20 0.34
DDR1 Q08345 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
DDR2 Q16832 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34
MAP3K20 Q9NYL2 1/20 0.34
MAP3K2 Q9Y2U5 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
HSP90AA1 P07900 1/20 0.33
TRPC1 P48995 1/20 0.33
STIM1 Q13586 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5060789 0.88 PTPN1 (0.41) GPR6MAPTTRPC3KDM4EALDH1A1
SCHEMBL5059312 0.83 KDM4E (0.39) GPR6MAPTTRPC3KDM4EALDH1A1
SCHEMBL1086640 0.79 GPR6 (0.40) GPR6MAPTTRPC3KDM4EALDH1A1
SCHEMBL5011733 0.76 EPHX2 (0.39) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL1086962 0.67 GPR6 (0.41) GPR6MAPTTRPC3CCR1PTPN1
SCHEMBL2858054 0.65 GPR6 (0.53) GPR6MAPTTRPC3KDM4EALDH1A1
SCHEMBL28696410 0.65 ALDH1A1 (0.76) GPR6MAPTTRPC3KDM4EALDH1A1
SCHEMBL2856010 0.64 MAPT (0.58) GPR6MAPTTRPC3KDM4EALDH1A1
SCHEMBL2064195 0.64 MAPT (0.76) GPR6MAPTTRPC3KDM4EALDH1A1
SCHEMBL2857536 0.64 TP53 (0.59) GPR6MAPTKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed