SCHEMBL5011733

SCHEMBL5011733

O=C1OC2(CCCCC2)N(C(=O)c2ccc(SC(F)(F)F)cc2)N1Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
PRKAB2 O43741 3/20 0.38
PRKAG1 P54619 3/20 0.38
PRKAA2 P54646 3/20 0.38
PRKAA1 Q13131 3/20 0.38
PRKAG3 Q9UGI9 3/20 0.38
PRKAG2 Q9UGJ0 3/20 0.38
PRKAB1 Q9Y478 3/20 0.38
HDAC1 Q13547 1/20 0.38
CHRM4 P08173 1/20 0.37
ADRB2 P07550 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
HIF1A Q16665 3/20 0.37
EPAS1 Q99814 3/20 0.37
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011835 0.80 CYP1A2 (0.43) HPGDPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL5056159 0.76 GPR6 (0.38) MEN1KMT2ASMN1; SMN2KDM4EALDH1A1
SCHEMBL1086650 0.74 EPHX2 (0.47) EPHX2MEN1HPGDTSHRKMT2A
SCHEMBL5011747 0.71 KCNK3 (0.40) HPGDKMT2ACYP3A4CYP2C9ALDH1A1
SCHEMBL5011879 0.69 KMT2A (0.38) MEN1HPGDTSHRKMT2ASMN1; SMN2
SCHEMBL5013344 0.68 CNR2 (0.38) MEN1HPGDTSHRKMT2ACYP3A4
SCHEMBL5012911 0.68 PPARG (0.36) HPGDTSHRKMT2AHIF1ACYP3A4
SCHEMBL5011651 0.68 CHRM2 (0.44) MEN1TSHRKMT2AADRB2SMN1; SMN2
SCHEMBL5015147 0.67 KMT2A (0.37) EPHX2MEN1TSHRKMT2AKDM4E
SCHEMBL1086092 0.64 RIPK1 (0.39) EPHX2MEN1KMT2ACHRM4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed