SCHEMBL5056804

SCHEMBL5056804

CCOC(=O)c1cc(Cl)c(=O)[nH]c1C.CCOC(=O)c1ccc(=O)[nH]c1C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
MAPT P10636 3/20 0.61
LMNA P02545 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
GAA P10253 2/20 0.57
POLB P06746 2/20 0.57
NPC1 O15118 1/20 0.57
PDE3B Q13370 3/20 0.53
PDE3A Q14432 3/20 0.53
CDK5 Q00535 2/20 0.47
CDK5R1 Q15078 2/20 0.47
KDM4E B2RXH2 4/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
BAZ2B Q9UIF8 1/20 0.43
BAZ2A Q9UIF9 1/20 0.43
CA12 O43570 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4881234 0.90 ALDH1A1 (0.73) ALDH1A1MAPTLMNAL3MBTL1GAA
SCHEMBL612717 0.86 ALDH1A1 (0.60) ALDH1A1MAPTLMNAL3MBTL1GAA
SCHEMBL18395324 0.80 TSHR (0.50) ALDH1A1MAPTLMNAL3MBTL1GAA
SCHEMBL9671945 0.77 ALDH1A1 (1.00) ALDH1A1MAPTLMNAL3MBTL1GAA
SCHEMBL4175783 0.75 PDE3B (0.60) ALDH1A1MAPTLMNAL3MBTL1GAA
SCHEMBL4876345 0.74 ALDH1A1 (0.76) ALDH1A1MAPTLMNAL3MBTL1GAA
SCHEMBL3593126 0.73 ALDH1A1 (0.49) ALDH1A1MAPTLMNAL3MBTL1GAA
SCHEMBL950017 0.73 ALDH1A1 (0.73) ALDH1A1MAPTLMNAL3MBTL1GAA
SCHEMBL4871436 0.73 GAA (1.00) ALDH1A1MAPTLMNAL3MBTL1GAA
SCHEMBL18796672 0.73 PDE3B (0.73) ALDH1A1MAPTLMNAL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904474-A1 NEW PYRIDINE ANALOGUES AstraZeneca AB (SE) 2008-04-02 EP disclosed
WO-2007008140-A1 NEW PYRIDINE ANALOGUES ASTRAZENECA AB (SE) 2007-01-18 WO disclosed