SCHEMBL5060050

SCHEMBL5060050

CCC(N)C1Cc2cccc(-c3cccnc3)c2O1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 7/20 0.39
CYP11B2 P19099 7/20 0.39
CYP19A1 P11511 3/20 0.39
PRKAB2 O43741 2/20 0.39
PRKAG1 P54619 2/20 0.39
PRKAA2 P54646 2/20 0.39
PRKAA1 Q13131 2/20 0.39
PRKAG3 Q9UGI9 2/20 0.39
PRKAG2 Q9UGJ0 2/20 0.39
PRKAB1 Q9Y478 2/20 0.39
CYP17A1 P05093 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP1A2 P05177 2/20 0.35
TDO2 P48775 1/20 0.35
PTGS2 P35354 1/20 0.34
DRD2 P14416 1/20 0.34
HTR7 P34969 1/20 0.34
MAOA P21397 1/20 0.34
KCNA5 P22460 1/20 0.34
MKNK1 Q9BUB5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595329 0.77 MAOA (0.47) CYP11B1CYP11B2CYP19A1CYP17A1CYP1A2
SCHEMBL4225039 0.77 PRKAB2 (0.59) CYP11B1CYP11B2CYP19A1PRKAB2PRKAG1
SCHEMBL5583580 0.77 PRKAB2 (0.37) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4595328 0.75 CYP11B1 (0.43) CYP11B1CYP11B2CYP19A1PRKAB2PRKAG1
SCHEMBL5141673 0.74 PRKAB2 (0.44) CYP11B1CYP11B2CYP19A1PRKAB2PRKAG1
SCHEMBL4232184 0.74 AQP1 (0.46) CYP11B1CYP11B2CYP19A1PRKAB2PRKAG1
SCHEMBL5077978 0.72 PRKAB2 (0.46) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4609187 0.70 PRKAB2 (0.42) CYP11B1CYP11B2PRKAB2PRKAG1PRKAA2
SCHEMBL14112685 0.70 PRKAB2 (0.46) CYP11B1CYP11B2CYP19A1PRKAB2PRKAG1
SCHEMBL14112652 0.70 PRKAB2 (0.46) CYP11B1CYP11B2CYP19A1PRKAB2PRKAG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871354-A1 TREATMENT OF PAIN Wyeth (US) 2008-01-02 EP disclosed
WO-2006116171-A1 TREATMENT OF PAIN WYETH (US) 2006-11-02 WO disclosed