SCHEMBL5067377

SCHEMBL5067377

CC(Cc1cccc(Cl)c1Cl)C(N)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 2/20 0.48
TAAR1 Q96RJ0 1/20 0.44
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
IDO1 P14902 2/20 0.43
ADA P00813 1/20 0.43
SLC6A2 P23975 3/20 0.41
SLC6A4 P31645 3/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP1A2 P05177 1/20 0.41
NFKB1 P19838 1/20 0.41
SLC6A3 Q01959 2/20 0.40
KCNH2 Q12809 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
GLA P06280 1/20 0.40
P2RX7 Q99572 2/20 0.39
CXCL8 P10145 1/20 0.39
PYGL P06737 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16973793 0.81 L3MBTL1 (0.42) IDO1CYP1A2ALDH1A1LMNA
SCHEMBL30962394 0.81 PNMT (0.50) PNMTTAAR1GRIN1GRIN2BIDO1
SCHEMBL18568286 0.80 PNMT (0.44) PNMTTAAR1GRIN1GRIN2BIDO1
SCHEMBL11434668 0.80 PNMT (0.44) PNMTTAAR1GRIN1GRIN2BIDO1
SCHEMBL8076310 0.77 PNMT (0.48) PNMTTAAR1IDO1SLC6A2SLC6A4
SCHEMBL3885817 0.77 PNMT (0.57) PNMTTAAR1IDO1SLC6A2SLC6A4
SCHEMBL18567935 0.77 PNMT (0.52) PNMTTAAR1IDO1SLC6A2SLC6A4
SCHEMBL13692532 0.77 PNMT (0.57) PNMTTAAR1IDO1SLC6A2SLC6A4
SCHEMBL5805934 0.77 PNMT (0.52) PNMTTAAR1IDO1SLC6A2SLC6A4
SCHEMBL8803316 0.76 MAOB (0.49) PNMTCYP3A4P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910272-A1 RENIN INHIBITORS Merck Frosst Canada Ltd. (CA) 2008-04-16 EP claimed
WO-2007009250-A1 RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2007-01-25 WO claimed