SCHEMBL506861

SCHEMBL506861

CCCCCCCCCCCCCCNC(=O)[C@H](CO)NCc1ccccc1O

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TLR2 O60603 2/20 0.53
NAAA Q02083 4/20 0.50
CA12 O43570 3/20 0.44
CA2 P00918 3/20 0.44
CA9 Q16790 3/20 0.44
EPHX1 P07099 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HTT P42858 1/20 0.42
MEN1 O00255 1/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506862 1.00 TLR2 (0.53) TLR2NAAACA12CA2CA9
SCHEMBL6241121 0.88 TLR2 (0.51) TLR2NAAACA12CA2CA9
SCHEMBL6936553 0.87 TLR2 (0.58) TLR2NAAAALDH1A1MEN1HPGD
SCHEMBL6936560 0.87 TLR2 (0.58) TLR2NAAAALDH1A1MEN1HPGD
SCHEMBL506094 0.87 TLR2 (0.52) TLR2NAAAEPHX1ALDH1A1HTT
SCHEMBL506095 0.87 TLR2 (0.52) TLR2NAAAEPHX1ALDH1A1HTT
SCHEMBL7224165 0.85 GRIA1 (0.53) TLR2
SCHEMBL6241805 0.85 NAAA (0.56) TLR2NAAACA12CA2CA9
SCHEMBL6934205 0.85 NAAA (0.56) TLR2NAAACA12CA2CA9
SCHEMBL6930474 0.85 NAAA (0.56) TLR2NAAACA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8853452-B2 Compounds, their syntheses, compositions, and methods to treat cancer THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2014-10-07 US disclosed
US-8853452-B2 Compounds, their syntheses, compositions, and methods to treat cancer THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2014-10-07 US disclosed
US-20120027844-A1 COMPOUNDS, THEIR SYNTHESES, COMPOSITIONS, AND METHODS TO TREAT CANCER XAVIER UNIVERSITY OF LOUISIANA (US) 2012-02-02 US disclosed
WO-2010093615-A2 COMPOUNDS, THEIR SYNTHESES, COMPOSITIONS, AND METHODS TO TREAT CANCER TULANE UNIVERSITY (US) 2010-08-19 WO disclosed
WO-2010093615-A2 COMPOUNDS, THEIR SYNTHESES, COMPOSITIONS, AND METHODS TO TREAT CANCER TULANE UNIVERSITY (US) 2010-08-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120027844-A1 COMPOUNDS, THEIR SYNTHESES, COMPOSITIONS, AND METHODS TO TREAT CANCER SGMS1, PHOSPHO1, MCL1 TLR2 4454/4885NAAA 987/4885CA12 2960/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.