SCHEMBL5072133

SCHEMBL5072133

CC(C(=O)OCCCN)(c1ccccc1)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 15/20 0.60
CHRM1 P11229 12/20 0.60
CHRM3 P20309 12/20 0.60
CHRM4 P08173 10/20 0.60
CHRM5 P08912 6/20 0.60
BCHE P06276 2/20 0.48
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10029779 0.85 CHRM2 (0.66) CHRM2CHRM1CHRM3CHRM4CHRM5
SCHEMBL15305877 0.79 CHRM2 (0.84) CHRM2CHRM1CHRM3CHRM4CHRM5
SCHEMBL28352271 0.78 CHRM2 (0.64) CHRM2CHRM1CHRM3CHRM4CHRM5
SCHEMBL29156932 0.78 CHRM2 (0.64) CHRM2CHRM1CHRM3CHRM4CHRM5
SCHEMBL8309422 0.77 CHRM2 (0.60) CHRM2CHRM1CHRM3CHRM4CHRM5
SCHEMBL31256699 0.76 CHRM2 (0.58) CHRM2CHRM1CHRM3CHRM4CHRM5
SCHEMBL30712480 0.76 ALDH1A1 (0.64) CHRM2CHRM1CHRM3CHRM4CHRM5
Aprofene SCHEMBL2354824 0.75 CHRM2 (1.00) CHRM2CHRM1CHRM3CHRM4CHRM5
SCHEMBL9588270 0.75 ALDH1A1 (0.68) CHRM2CHRM1CHRM3CHRM4CHRM5
SCHEMBL28555859 0.75 CHRM2 (0.53) CHRM2CHRM1CHRM3CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012055018-A1 THERAPEUTIC COMPOSITIONS FOR DIABETIC SYMMETRICAL POLYNEUROPATHY UNIVERSITY OF MANITOBA (CA) 2012-05-03 WO disclosed