SCHEMBL5072230

SCHEMBL5072230

CC(=O)Nc1cc(-c2ccccc2)c([N+](=O)[O-])cc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
MAPT P10636 3/20 0.45
NPSR1 Q6W5P4 2/20 0.45
PKM P14618 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
HTT P42858 2/20 0.44
PDE7A Q13946 1/20 0.44
TDP1 Q9NUW8 2/20 0.43
HDAC1 Q13547 2/20 0.43
KDM4E B2RXH2 1/20 0.43
APOBEC3A P31941 1/20 0.43
GFER P55789 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC2 Q92769 1/20 0.42
RXFP1 Q9HBX9 1/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26631727 0.81 ALDH1A1 (0.54) ALDH1A1MAPTNPSR1PKMHTT
SCHEMBL30691972 0.81 ALDH1A1 (0.54) ALDH1A1MAPTNPSR1PKMHTT
SCHEMBL5069542 0.80 MAPT (0.54) ALDH1A1MAPTNPSR1PKML3MBTL1
SCHEMBL20096855 0.79 MAPT (0.45) ALDH1A1MAPTNPSR1PKML3MBTL1
SCHEMBL6378334 0.78 HTT (0.49) ALDH1A1MAPTNPSR1PKML3MBTL1
SCHEMBL11638099 0.77 POLB (0.48) ALDH1A1MAPTNPSR1PKML3MBTL1
SCHEMBL5068702 0.77 ALDH1A1 (0.56) ALDH1A1MAPTPDE7ATDP1CYP3A4
SCHEMBL23579968 0.76 MAPT (0.47) ALDH1A1MAPTNPSR1PKML3MBTL1
SCHEMBL7653533 0.75 MAPT (0.55) ALDH1A1MAPTNPSR1PKML3MBTL1
SCHEMBL2645986 0.75 ABCB1 (0.66) ALDH1A1MAPTNPSR1HTTHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1319231-A4 PROGRAMMABLE MOLECULAR DEVICE UNIV WM MARSH RICE (US) 2008-11-19 EP disclosed
EP-1319231-A1 PROGRAMMABLE MOLECULAR DEVICE Wm. MARSH RICE UNIVERSITY (US) 2003-06-18 EP disclosed
US-20030058697-A1 Programmable molecular device NAVY, SECRETARY OF THE, UNITED STATES OF AMERICA OFFICE OF NAVAL RESEARCH 2003-03-27 US disclosed
WO-2002009117-A1 PROGRAMMABLE MOLECULAR DEVICE WM. MARSH RICE UNIVERSITY (US) 2002-01-31 WO disclosed